首页 » Biovector稳定细胞株库|外源蛋白过表达稳定细胞株列表1,GPCR & 离子通道稳定细胞系

Biovector稳定细胞株库|外源蛋白过表达稳定细胞株列表1,GPCR & 离子通道稳定细胞系

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Biovector稳定细胞株库

外源蛋白过表达稳定细胞株列表1



母细胞外源基因
HEK293ADORA1/Ga15/HEK293
CHOADRA1A/CHO
CHOADRA1B/CHO
HEK293ADRB2/bla(b)+beta-arrestin2/bla(b)/HEK293
HEK293AGTR1/Ga16/HEK293
CHOalpha1a/CHO
HEK293alpha1b/HEK293
HEK293alpha1DAR-Ga16/HEK293
HEK293AVPR2/Ga16/HEK293
CHOB2/Ga15/CHO
CHOBB1/CHO
HEK293BDKRB1/HEK293
HEK293beta2AR/Ga16/HEK293
CHOCB1/Ga16/CHO
CHOCB2/Ga16/CHO
CHOCCKA/Ga15/CHO
CHOCCKB/CHO
CHOCCR1/Ga16/CHO
HEK293CCR2/Ga16/HEK293
CHOCCR5-Ga16/CHO
CHOCXCR2/Ga16/CHO
CHOCXCR4/Ga16/CHO
HEK293DRD1/Ga16/HEK293
HEK293DRD2/Ga16/HEK293
HEK293DRD5/Ga16/HEK293
CHOEDNRA/CHO
CHOEDNRB/CHO
HEK293GCGR/Ga16/HEK293
CHOGL1P-Ga16/CHO
HEK293GLP1R/Ga16/HEK293
HEK293GLP2R/Ga16/HEK293
HEK293H1/HEK293
CHOH2/Ga15/CHO
CHOH3/Ga15/CHO
CHOH4/Ga15/CHO
HEK293hERG
CHOM1/CHO
HEK293M2-Ga16/HEK293
HEK293M3/HEK293
HEK293M4/Ga16/HEK293
CHOM5/CHO
HEK293MC1R-Ga16/HEK293
HEK293MC3R/Luc/HEK293
HEK293MC4R/Luc/HEK293
HEK293MOR/Ga16/HEK293
HEK293NPY1R-Ga16/HEK293
HEK293NPY2R-Ga16/HEK293
HEK293NPY4R-Ga16/HEK293
HEK293NPY5R-Ga16/HEK293
HEK293OX1/HEK293
CHOOX2/CHO
CHOTRPA1
HEK293TRPC1
HEK293TRPC6
CHOTRPM2
CHOTRPM8
CHOTRPV1
CHOTRPV4
ADORA1/Ga15/HEK293稳定表达细胞株
ADRA1A/CHO稳定表达细胞株
ADRA1B/CHO稳定表达细胞株
ADRB2/bla(b)+beta-arrestin2/bla(b)/HEK293稳定表达细胞株
AGTR1/Ga16/HEK293稳定表达细胞株
alpha1a/CHO稳定表达细胞株
alpha1b/HEK293稳定表达细胞株
alpha1DAR-Ga16/HEK293稳定表达细胞株
AVPR2/Ga16/HEK293稳定表达细胞株
B2/Ga15/CHO稳定表达细胞株
BB1/CHO稳定表达细胞株
BDKRB1/HEK293稳定表达细胞株
beta2AR/Ga16/HEK293稳定表达细胞株
CB1/Ga16/CHO稳定表达细胞株
CB2/Ga16/CHO稳定表达细胞株
CCKA/Ga15/CHO稳定表达细胞株
CCKB/CHO稳定表达细胞株
CCR1/Ga16/CHO稳定表达细胞株
CCR2/Ga16/HEK293稳定表达细胞株
CCR5-Ga16/CHO稳定表达细胞株
CXCR2/Ga16/CHO稳定表达细胞株
CXCR4/Ga16/CHO稳定表达细胞株
DRD1/Ga16/HEK293稳定表达细胞株
DRD2/Ga16/HEK293稳定表达细胞株
DRD5/Ga16/HEK293稳定表达细胞株
EDNRA/CHO稳定表达细胞株
EDNRB/CHO稳定表达细胞株
GCGR/Ga16/HEK293稳定表达细胞株
GL1P-Ga16/CHO稳定表达细胞株
GLP1R/Ga16/HEK293稳定表达细胞株
GLP2R/Ga16/HEK293稳定表达细胞株
H1/HEK293稳定表达细胞株
H2/Ga15/CHO稳定表达细胞株
H3/Ga15/CHO稳定表达细胞株
H4/Ga15/CHO稳定表达细胞株
hERG稳定表达细胞株
M1/CHO稳定表达细胞株
M2-Ga16/HEK293稳定表达细胞株
M3/HEK293稳定表达细胞株
M4/Ga16/HEK293稳定表达细胞株
M5/CHO稳定表达细胞株
MC1R-Ga16/HEK293稳定表达细胞株
MC3R/Luc/HEK293稳定表达细胞株
MC4R/Luc/HEK293稳定表达细胞株
MOR/Ga16/HEK293稳定表达细胞株
NPY1R-Ga16/HEK293稳定表达细胞株
NPY2R-Ga16/HEK293稳定表达细胞株
NPY4R-Ga16/HEK293稳定表达细胞株
NPY5R-Ga16/HEK293稳定表达细胞株
OX1/HEK293稳定表达细胞株
OX2/CHO稳定表达细胞株
TRPA1稳定表达细胞株
TRPC1稳定表达细胞株
TRPC6稳定表达细胞株
TRPM2稳定表达细胞株
TRPM8稳定表达细胞株
TRPV1稳定表达细胞株
TRPV4稳定表达细胞株
Amylin 3受体表达细胞株Amylin 3 ReceptorBiovector™ Amylin 3 Receptor
大麻素受体表达细胞株Cannabinoid ReceptorBiovector™ Cannabinoid Receptor
细胞趋化因子(C-C) 受体2B表达细胞株Chemokine (C-C) Receptor 2BBiovector™ Chemokine (C-C) Receptor 2B
细胞趋化因子(C-X-C motif)受体4表达细胞株Chemokine (C-X-C motif) Receptor 4Biovector™ Chemokine (C-X-C motif) Receptor 4
多巴胺受体1表达细胞株Dopamine Receptor 1 (DRD1)Biovector™ Dopamine Receptor 1 (DRD1)
胰高血糖样受体1表达细胞株Glucagon-like Receptor 1 (GLP1R)Biovector™ Glucagon-like Receptor 1 (GLP1R)
阿片样受体1表达细胞株Opiate Receptor-like 1 (ORL1Biovector™ Opiate Receptor-like 1 (ORL1


GPCR & 离子通道稳定细胞系








NTCC Biovector  Inc.为客户提供种类丰富的GPCR和离子通道稳定细胞系。凭借密码子优化和载体设计的专利技术,我们成功克服了细胞表面功能蛋白表达水平低的难题。NTCC Biovector  Inc.所有的细胞系均针对钙流检测、FRET检测和化学发光检测法中的信号窗口(S/B ratio)进行了优化,并通过了16次传代的稳定性验证。








主要特性








细胞表面功能蛋白表达水平高




实验结果可靠,可重现




所有的离子通道稳定细胞系都通过手动膜片钳和Qpatch验证




多种功能参数可供选择








产品信息




受体家族

受体

细胞系

产品编号

5-Hydroxytryptamine receptor

5-HT1A/HTR1A

CHO-K1/5-HT1A/Gα15

NTCC00330

5-HT2A/HTR2A

CHO-K1/5-HT2A

NTCC00251

5-HT2B/HTR2B

CHO-K1/5-HT2B

NTCC00249

5-HT2C/HTR2C

CHO-K1/5-HT2C

NTCC00253

5-HT2C/HTR2C

HEK 293/5-HT2C

NTCC00319

HTR4

CHO-K1/5-HT4/Gα15

NTCC00444

HTR7

293/5-HT7/CRE-Luc

NTCC00423

Acetylcholine receptor (muscarinic)

M1/CHRM1

CHO-K1/M1

NTCC00185

M2/CHRM2

CHO-K1/M2/Gα15

NTCC00258

M3/CHRM3

CHO-K1/M3

NTCC00259

M4/CHRM4

CHO-K1/M4/Gα15

NTCC00238

M5/CHRM5

CHO-K1/M5

NTCC00186

Adenosine receptor

ADORA1

CHO-K1/ADORA1/Gα15

NTCC00324

ADORA1

293/ADORA1/Gα15

NTCC00255

ADORA2a

CHO-K1/ADORA2A/Gα15

NTCC00246

ADORA2B

CHO-K1/ADORA2B/Gα15

NTCC00329

ADORA3

CHO-K1/ADORA3/Gqi5

NTCC00464

Adrenoceptors

ADRB3

293/ADRB3/CRE-Luc

NTCC00335

ADRA1B

CHO-K1/ADRA1B

NTCC00260

ADRA1D

CHO-K1/ADRA1D

NTCC00340

ADRA2A

CHO-K1/ADRA2A/Gα15

NTCC00281

ADRA2B

CHO-K1/ADRA2B/Gqi5

NTCC00454

ADRA2C

CHO-K1/ADRA2C/Gα15

NTCC00252

ADRB1

CHO-K1/ADRB1/Gα15

NTCC00269

ADRA1A

CHO-K1/ADRA1A

NTCC00225

Angiotensin receptor

AT1

HEK 293/AT1

NTCC00458

AT1

293T/AT1

NTCC00448

Apelin receptor

AGTRL1

CHO-K1/AGTRL1/Gα15

NTCC00245

Bile acid receptor

GPBAR1

CHO-K1/GPBAR1SatbleCellLine

NTCC00432









受体家族

受体

细胞系

产品编号

Bombesin receptor

BB1

CHO-K1/BB1

NTCC00254

BB2/GRPR

CHO-K1/BB2

NTCC00182

BB3/BRS3

CHO-K1/BB3

NTCC00183

Bradykinin receptor

B2

CHO-K1/B2/Gα15

NTCC00184

Calcitonin

AMY1

CHO-K1/AMY1/Gα15

NTCC00475

Calcitonin receptor

CALCR/CT

CHO-K1/CT/Gα15

NTCC00320

Calcium-sensing receptor

CASR

CHO-K1/CASR

NTCC00434

Cannabinoid receptor

CNR1/CB1

CHO-K1/CB1/Gα15

NTCC00299

CB2

CHO-K1/CB2

NTCC00433

Chemerin receptor

CMKLR1

CHO-K1/CMKLR1/Gα15

NTCC00301

Chemokine receptor

CCR1

CHO-K1/Gα15/CCR1   New

NTCC00522

CCR5

CHO-K1/Gα15/CCR5   New

NTCC00523

CXCR1/IL8RA

CHO-K1/Gα15/CXCR1   New

NTCC00524

CXCR3

CHO-K1/Gα15/CXCR3   New

NTCC00525

CXCR5/BLR1

CHO-K1/Gα15/CXCR5   New

NTCC00526

Cholecystokinin receptor

CCKA/CCKAR

CHO-K1/CCKA/Gα15

NTCC00271

CCKB/CCKBR

CHO-K1/CCKB

NTCC00154

Class A orphan

GPR68/OGR1

CHO-K1/GPR68/Gα15

NTCC00439

MRGPRX2

CHO-K1/MRGPRX2

NTCC00425

Complement peptide receptor

C5a/C5AR1

CHO-K1/C5a/Gα15

NTCC00327

Corticotropin releasing factor receptor

CRF1/CRHR1

CHO-K1/CRF1/Gα15

NTCC00343

CRF2

CHO-K1/CRF2/Gα15

NTCC00208

Dopamine receptor

D2

CHO-K1/D2/Gα15

NTCC00152

D5

CHO-K1/D5/Gα15

NTCC00322

D1/DRD1

CHO-K1/D1

NTCC00247

D2(Short)

CHO-K1/D2s/Gα15

NTCC00274

Endothelin receptor

ETA/EDNRA

CHO-K1/EDNRA

NTCC00149

ETB/EDNRB

CHO-K1/EDNRB

NTCC00150

Formylpeptide receptor

FPR1

CHO-K1/FPR1/Gα15

NTCC00429

Free fatty acid receptor

FFA2

CHO-K1/FFA2/Gα15

NTCC00437

GPR40/FFA1

CHO-K1/FFA1/Gα15

NTCC00273

返回顶部








受体家族

受体

细胞系

产品编号

Galanin receptor

GAL1/GALR1

CHO-K1/GAL1/Gα15

NTCC00277

GAL2/GALR2

CHO-K1/GAL2

NTCC00209

Glucagon receptor

GHRHR

293/GHRH/Gα15

NTCC00314

GLP-1/GLP1R

CHO-K1/GLP1/Gα15

NTCC00451

GLP-2/GLP2R

CHO-K1/GLP2/Gα15

NTCC00307

GCGR

CHO-K1/GCGR/Gα15

NTCC00345

GCGR

HEK 293/GCGR/Gα15

NTCC00422

SCTR

CHO-K1/SCTR/Gα15

NTCC00326

GIPR

CHO-K1/GIP/Gα15

NTCC00486

Gonadotropin releasing hormone receptor

GNRHR

CHO-K1/GNRHR/Gα15

NTCC00426

Growth hormone releaseing peptides receptor

GHSR

CHO-K1/GHSR

NTCC00189

Histamine receptor

H1/HRH1

293/H1

NTCC00131

H2/HRH2

CHO-K1/H2/Gα15

NTCC00306

H3/HRH3

CHO-K1/H3/Gα15

NTCC00331

H4/HRH4

CHO-K1/H4/Gα15

NTCC00289

Hydroxycarboxlic acid receptor

GPR109A

CHO-K1/NIACR1/Gα15

NTCC00428

Kisspeptin receptor

KiSS1/GPR54

CHO-K1/KiSS1

NTCC00190

Leukotriene receptor

FPRL1

CHO-K1/FPRL1/Gα15

NTCC00305

CysLT1

CHO-K1/CysLT1/Gα15

NTCC00462

LTB4R

CHO-K1/LTB4/Gα15

NTCC00435

Lysophospholipid receptor

EDG4/LAP2

RH7777/EDG4

NTCC00463

Melanin concentrating hormone receptor

MCH1/GPR24

293/MCH1

NTCC00211

MCH2/GPR145

CHO-K1/MCH2

NTCC00280

Melanocortin receptor

MC2

CHO-K1/MC2/Gα15

NTCC00336

MC3

CHO-K1/MC3/Gα15

NTCC00242

MC3

293/MC3/CRE-Luc

NTCC00337

MC4

CHO-K1/MC4/Gα15

NTCC00272

MC5

CHO-K1/MC5/Gα15

NTCC00243

Melatonin receptor

MTNR1A

CHO-K1/MT1/Gα15

NTCC00424

MT2/MTNR1B

CHO-K1/MT2/Gα15

NTCC00312

Metabropic glutamate receptor

mGlu2/GRM2

CHO-K1/GRM2/Gα15

NTCC00427

Motilin receptor

MTLR/MLNR

CHO-K1/MTLR/Gα15

NTCC00347

返回顶部








受体家族

受体

细胞系

产品编号

Neuromedin receptor

NMU2

293T/NMU2

NTCC00244

NMU1/GPR66

CHO-K1/NMU1

NTCC00191

Neuropeptide S receptor

NPS1b

CHO-K1/NPS1b/Gα15

NTCC00344

NPSR1

CHO-K1/NPS1a/Gα15

NTCC00338

Neuropeptide Y receptor

NPY2

CHO-K1/NPY2/Gqi5

NTCC00460

NPY4R

CHO-K1/NPY4/Gα15

NTCC00237

Neurotensin receptor

NTS1/NT1

CHO-K1/NTS1

NTCC00194

Opioid & opioid-like receptor

OPRD1

CHO-K1/OPRD1/Gα15

NTCC00323

OPRK1

CHO-K1/OPRK1/Gα15

NTCC00290

OPRM1

CHO-K1/OPRM1/Gα15

NTCC00304

OPRL1

CHO-K1/OPRL1/Gα15

NTCC00447

Orexin receptor

OX1

CHO-K1/OX1

NTCC00224

OX2

CHO-K1/OX2

NTCC00316

P2Y receptor

P2Y1

1321N1/P2Y1

NTCC00250

P2Y2

1321N1/P2Y2

NTCC00318

P2Y4

1321N1/P2Y4

NTCC00297

P2Y6

1321N1/P2Y6

NTCC00346

P2Y11

1321N1/P2Y11

NTCC00298

P2Y12

1321N1/P2Y12/Gα15

NTCC00261

Parathyroid hormone receptor

PTH1/PTHR1

CHO-K1/PTH1/Gα15

NTCC00315

PTH2/PTHR2

293/PTH2/CRE-Luc

NTCC00270

Peptide P518 receptor

QRFP/GPR103

CHO-K1/GPR103/Gα15

NTCC00321

Platelet activating factor receptor

PAFR/PTAFR

CHO-K1/PTAFR

NTCC00262

Prolactin releasing peptide receptor

PRLHR

CHO-K1/PRLHR

NTCC00341

Prostanoid receptor

DP2

CHO-K1/DP2/Gα15

NTCC00436

EP1/PTGER1

293/EP1

NTCC00228

EP2/PTGER2

CHO-K1/EP2/Gα15

NTCC00311

FP/PTGFR

293/FP/Gα15

NTCC00155

IP1/PTGIR

CHO-K1/IP1/Gα15

NTCC00310

TP/TBXA2R

293/TP

NTCC00309

PTGDR/DP1

CHO-K1/DP1/Gα15

NTCC00453

Proteinase-activated receptor

PAR2

CHO-K1/PAR2/Gα15

NTCC00446

PAR4/F2RL3

CHO-K1/PAR4

NTCC00206









受体家族

受体

细胞系

产品编号

Somatostatin receptor

SST1

CHO-K1/SST1/Gqi5

NTCC00473

SST2/SSTR2

CHO-K1/SST2/Gα15

NTCC00325

SST3

CHO-K1/SST3/Gα15

NTCC00285

SST4/SSTR4

CHO-K1/SST4/Gα15

NTCC00334

SST5/SSTR5

CHO-K1/SST5/Gα15

NTCC00286

Tachykinin receptor

NK1/TACR1

CHO-K1/NK1

NTCC00199

NK2/TACR2

CHO-K1/NK2

NTCC00200

NK3/TACR3

CHO-K1/NK3

NTCC00201

Thyrtropin releasing hormone receptor

TRH1/TRHR

CHO-K1/TRH1

NTCC00202

Urotensin receptor

UTR2

CHO-K1/UT2/Gα15

NTCC00339

Vasopressin and oxytocin receptor

OT/OXTR

CHO-K1/OXTR

NTCC00195

V1B

CHO-K1/V1B

NTCC00205

V2

CHO-K1/V2/Gα15

NTCC00170

VIP, Vasoactive intestinal polypeptide receptor 2

PAC1

CHO-K1/PAC1/Gα15

NTCC00203

VIP, Vasoactive intestinal polypeptide receptor 3

VPAC2

CHO-K1/VPAC2/Gα15

NTCC00226

VIP, Vasoactive intestinal polypeptide receptor 4

VPAC1/VIP1

CHO-K1/VPAC1/Gα15

NTCC00342

Control

\

CHO-K1/CRE/Luc

NTCC00187

\

CHO-K1/Gα15

NTCC00257

\

CHO-K1/Gqi5

NTCC00455










I.GPCRcelllines



No.

Family

Receptor

Species

CellLine

1




5-Hydroxytryptamine

5-HT1A

human

HEK293/Ga16/HTR1A

2

5-HT2A

human

HEK293/HTR2A

3

5-HT2B

human

HEK293/HTR2B

4

5-HT2C

human

HEK293/Ga16/HTR2C

5

5-HT6

human

HEK293/5HT6

6

5-HT7

human

HEK293/5HT7

7






Adenosine

ADORA1

human

HEK293/Ga15/ADORA1

8


ADORA2A

human

HEK293/ADORA2A

9

mouse

HEK293/mADORA2A

10



ADORA3

human

CHO-K1/ADORA3/β-Arrestin

11

human

CHO-K1/ADORA3

12

mouse

CHO-K1/mAdora3

13

human

HEK293/G15/ADORA3

14

ADORA2B

human

HEK293/G15/ADORA2B

15








Adrenergic

Alpha-1A

human

HEK293/α1A

16

Alpha-1B

human

HEK293/α1B

17

Alpha-1D

human

HEK293/α1D

18


Alpha-2A

human

CHO-K1/Ga15/α2A

19

human

HEK293/Ga16/α2A

20

Alpha-2C

human

HEK293/Ga15/α2C

21



β2



human

HEK/beta 2/β-lactamasefragmentB/β-arrestin  fused

lactamaseA

22

HEK/CRE-GFP/β2

23

β3

human

HEK293/beta  3

24

Angiotensin

AT1

human

HEK293/Ga15/AT1

25

Bile acid

GPR131(TGR5)

human

CHO-K1/TRE/TGR5

26

Bombesin

BB3

human

HEK293/Ga15/BB3

27


Bradykinin

B1

human

HEK293/Ga15/B1

28

B2

human

HEK293/Ga15/B2

29

Calcitonin

CTR

human

CHO-K1/CTR1

30

Cannabinoid

CB2

human

HEK293/Ga15/CB2

31

Chemokine

CXCR1

human

HEK293/CXCR1



Page 1of5



32


CXCR2

human

HEK293/CXCR2

33

CCR4

human

HEK293/CCR4R

34

CCR6

human

HEK293/CCR6R

35


Cholecystokinin

CCKA

human

HEK293/CCK1R

36

CCKB

human

HEK293/CCK2R

37

Corticotropin-Releasing

hormone


CRHR2


human


HEK293/CRHR2

38




Dopamine

D1

human

HEK293/D1R/CRE/βla

39

D2L

human

HEK293/Ga15/D2RL

40

D2S

human

HEK293/Ga15/D2RS

41

D3

human

HEK293/Ga15/D3R

42

D4

human

HEK293/Ga15/D4R

43

D5

human

HEK293/D5R/CRE/βla

44


Endothelin

ETA

human

HEK293/ETA

45

ETB

human

HEK293/ETB

46


Free FattyAcid

GPR40

human

HEK293/GPR40

47

GPR119

human

LVIP/GPR119/CRE-b-gal

48

GPR120

human

HEK293/NFAT/bla/GPR120

49


Galanin

GALR1

human

HEK293/Ga16/GALR1

50

GALR2

human

CHO-K1/GALR2

51

Ghrelin

GHSR1a

human

HEK293/GHSR1a

52


Glucagon


GCGR

human

HEK293/Ga15/GCGR

53

human

HEK293/GCGR/CRE-Luc

54

GLP-1

human

HEK293/GLP1R/CRE-Luc

55

Gonadotrophin-releasinghormone


GRH


human


HEK293/GnRHR/NFAT/bla

56






Histamine

H1

human

HEK293/H1R/NFAT/bla

57

H2

human

HEK293/H2R/CRE/Luc

58


H3

human

HEK293/Ga15/H3R

59

human

HEK293/H3R/CRE-luc/Go2

60

human

H3R/SK-N-MC/CRE-b-gal

61


H4

human

HEK293/H4R/G16

62

human

SK-N-MC/H4R/CRE-b-gal

63

mouse

SK-N-MC/mH4R/CRE-b-gal

64


Melanin-ConcentratingHormone


MCH1

human

HEK293/huMCHR1

65

Rat

HEK293/rMCHR1

66

MCH2

human

HEK293/MCHR2

67



Melanocortin

MC1

human

HEK293/CRE-luc/MC1R

68

MC2

human

HEK293/CRE-luc/MC2R

69

MC3

human

HEK293/CRE-luc/MC3R

70

MC4

human

HEK293/Ga15/MC4R



71



human

HEK293/MC4R/CRE-GFP

72

MC5

human

HEK293/MC5R

73


Melatonin

MT1A

human

HEK293/G15/MT1A

74

MT1B

human

HEK293/G15/MT1B

75







Metabotropic  Glutamate


mGluR1

human

HEK293/humGluR1

76

human

CHO-K1/mGluR1

77

mGluR2

human

HEK293/Ga16/mGluR2

78

mGluR3

human

HEK293/Ga16/EAAC1/mGluR3

79

mGluR4

human

HEK293/Ga15/mGluR4

80


mGluR5

human

HEK293/mGluR5a

81

rat

HEK293/ratmGluR5

82

mGluR6

human

HEK293/Ga15/mGluR6

83

mGluR7

human

HEK293/Ga15/EAAC1/mGluR7

84

mGluR8

human

HEK293/Ga15/EAAC1/mGluR8

85

Mas-related  genes (Mrgs)

MrgD

human

CHO-K1/MrgD

86






Muscarinic


M1


human

HEK293/M1

87

CHO-K1/M1

88

U2OS/M1/NFATc1-EGFP

89


M2


human

CHO-K1/M2

90

CHO-K1/M2/PKAcat-EGFP

91


M3


human

HEK293/M3

92

CHO-K1/M3

93

M4

human

CHO-K1/Gα15/M4

94

M5

human

CHO-K1/M5

95

NeuromedinU

NMU1

human

HEK293/Ga15/NMU1R

96


Neuropeptide  FF


NPFFR 1

human

HEK293/NPFF1/CRE/luc

97

human

HEK293/Ga16/NPFF1

98

human

HEK293/G16/NPFF1/NFAT/blx

99


Neuropeptide  Y

NPY1

human

HEK293/Ga15/NPY1R

100

NPY2

human

HEK293/Ga15/NPY2R

101




Opioid

OPRD

human

HEK293/OPRD

102

OPRL1

human

HEK293/Ga15/OPRL1

103

OPRL1

human

CHO-K1/OPRL1

104

OPRK

human

CHO-K1/OPRK

105

OPRM

human

CHO-K1/OPRM

106

Orexin

OX1

human

HEK293/Ga15/OX1

107




OrphanReceptor

GPR3

human

HEK293/GPR3

108


GPR6

human

HEK293/GPR6/TREx

109


rat

HEK293/rGPR6 transient

assay

110

GPR12

human

HEK293/GPR12 transient







assay

111

GPR139

human

HEK293/GPR139

112

GPR142

human

HEK293/GPR142

113

GPR142

mouse

HEK293/mGPR142

114


GPR183

human

SK-N-MC/CREGPR183

115

human

HEK293  arrestin GPR183

116

mGPR48

mouse

HEK293/mGPR48/Topflash

117


Parathyroid  Hormone


PTHR 1

human

HEK293/PTHR1/CRE/bla

118

human

HEK293/PTHR1/CRE-GFP

119

PTHR 2

human

HEK293/PTHR2/CRE/bla

120

Platelet-activatingfactor

PAFR

human

HEK293/PAFR/NFAT/bla

121


Protease-activatedreceptors (thrombin)

PAR1

human

HEK293/Ga15/PAR1

122

PAR2 /F2RL1

human

HEK293/Ga15/PAR2

123

PAR4

human

HEK293/Ga15/PAR4

124




Somatostatin

sst1

human

HEK293/Ga15/sst1

125

sst2

human

HEK293/Ga15/sst2

126

sst3

human

HEK293/Ga15/sst3

127

sst4

human

HEK293/Ga15/sst4

128

sst5

human

HEK293/Ga15/sst5

129



Tachykinin

Substance

P/TACR1


human


HEK293/SPR

130

NK2

human

HEK293/NK2R

131

NK3

human

HEK293/Ga15/NK3R

132

Urotensin

UTR2

human

HEK293/Ga15/UTR2

133


Vasopressin


V1A

Cynomolgus

CHO-K1/V1A802

134

human

CHO-K1/V1A

135

V1B

human

CHO-K1/V1B



II.Ion channelcelllines


No.

Family

Ionchannel

Species

CellLine


1

4TMpotassiumchannelTREK1 (K2p2.1)


TREK1  (K2p2.1)


human


CHO-K1/TREK1

2



ATP-gated purinergicreceptor

P2RX1

human

HEK293/P2RX1

3

P2RX2

human

HEK293/P2RX2

4

P2RX4

human

HEK293/P2RX4

5

ratP2X4

rat

1321N1/rP2RX4

6

P2RX7

human

HEK293/P2RX7

7

Glycine  receptor

GLRα1/βa

human

CHO-K1/GLRα1/βa



8


GlyRα2

human

CHO-K1/GlyRα2

9

GLRα3a

human

CHO-K1/GLRα3a


10

Nicotine acetycholine

receptor

Alpha-4 beta-2

nicotinic receptor


human

CHO-K1/α4β2 nicotinic

receptor

11

Serotonin  receptor

5-HT3

human

CHO-K1/5-HT3

12





Transientreceptorpotentialchannel

TRPA1

human

HEK293/TRPA1

13

TRPM8

human

HEK293/TRPM8

14

TRPV1

human

HEK293/TRPV1

15

RatTRPV1

rat

HEK293/rTRPV1

16

TRPV2

human

HEK293/TRPV2

17

TRPV3

human

HEK293/TRPV3

18

TRPV4

human

HEK293/TRPV4

19

TRPV6

human

HEK293/TRPV6

20



Voltage-gated potassiumchannel

hERG

human

HEK293/hERG

21


KCNA5

human

HEK293/KCNA5

22

human

CHO-K1/KCNA5

23

KvLQT1/minK

human

CHO-K1/KvLQT1/minK


24

Voltage-gated sodium

channel


NaV1.8


human


CHO-K1/NaV1.8


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